B7-33
Muscle/RecoveryRelaxin-2 analog / researchEmerging
Single-chain relaxin-2 analog designed at Monash University as an RXFP1 agonist for anti-fibrotic and vasodilatory research. Preclinical; not FDA-approved.
For research use only.
Key Facts
- CAS
- โ
- Molecular Weight (MW)
- ~5 kDa
- Half-life
- Short; stabilized vs native relaxin-2
- Unit
- mcg
- Administration Route
- โ
- Frequency
- โ
- Last updated
- 8/23/2026
- Targets
- RXFP1 (relaxin family peptide receptor 1)
Overview
Single-chain relaxin-2 analog designed at Monash University as an RXFP1 agonist for anti-fibrotic and vasodilatory research. Preclinical; not FDA-approved.
Protocol
- Dosage Range
- Per research protocol
- Frequency
- โ
- Cycle
- โ
- Administration Route
- โ
- Reconstitution Guide
- โ
Science
Mechanism of Action
Minimized relaxin-2 analog that activates RXFP1, promoting vasodilation, extracellular-matrix remodeling, and anti-fibrotic signaling in heart and kidney models.
Targets
RXFP1 (relaxin family peptide receptor 1)
Studies
- B7-33 single-chain relaxin analogโ Journal/year not available
Benefits
Anti-fibrotic researchVasodilatory RXFP1 models
Potential Side Effects
- No established human dose
- Hypotension theoretical
References
- PMID 25589618External link ยท Year โ