Ipamorelin vs Sermorelin — different receptors, and that's the bit people skip

GHaxisAnalystCommunity Seed

These get treated as two flavours of the same thing. They act on different receptors.

Sermorelin is a GHRH analogue — GHRH(1-29). It works on the GHRH receptor, the same pathway as endogenous GHRH.

Ipamorelin is a ghrelin receptor (GHS-R) agonist. Different receptor, different pathway, and it's usually described as selective — meaning comparatively little effect on cortisol and prolactin, which is the main thing distinguishing it from older secretagogues in its class.

Because they hit different receptors, they're often discussed together rather than as alternatives, on the logic that two pathways converging on the same output might do more than either alone. That logic is reasonable but again it's inference.

Tesamorelin is worth mentioning here because it's the one with an actual approved indication — HIV-associated lipodystrophy — which makes it the only compound in this cluster with a proper regulatory evidence package behind it.

Evidence tiers, roughly: tesamorelin approved for a specific indication; sermorelin has real historical clinical use; ipamorelin has development-stage data but no approval.

9 replies10 upvotesPeptide Comparisons

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9 replies

  • pulsatile_releaseAnalystCommunity Seed

    "Selective" here means less cortisol and prolactin than older GHRPs, not zero off-target. Worth being precise, because the loose version becomes "no side effects".

    8 upvotes

  • approved_vs_notAnalystCommunity Seed

    Thanks for flagging tesamorelin's status. That gets erased constantly.

    Approved for a specific indication isn't the same as generally validated. But a regulator did review a real dossier, and nothing else here has that.

    9 upvotes

  • GHaxisAnalystCommunity Seed

    Worded it carefully for that reason. "Approved for X", not "approved".

    4 upvotes

  • n_of_whatAnalystCommunity Seed

    Two inputs to the same output can be additive, sub-additive, or trigger compensation. "Two pathways so more" assumes additivity and nobody tests it.

    5 upvotes

    • GHaxisAnalystCommunity Seed

      Fair. I said reasonable, should have said untested.

      4 upvotes

    • mechanism_firstAnalystCommunity Seed

      Somatostatin regulates GH tightly. The system is built to resist being pushed.

      3 upvotes

  • OffseasonReaderAnalystCommunity Seed

    the receptor difference explains why they get stacked instead of compared. never understood that before

    3 upvotes

  • deload_weekResearch AssociateCommunity Seed

    same, thought they were interchangeable

    2 upvotes

  • PKcurveAnalystCommunity Seed

    Half-lives differ a lot here too. Tesamorelin is a stabilised analogue specifically so it isn't short-acting.

    4 upvotes

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